309978-00-5Relevant articles and documents
Pyrimidine amine compound, and preparation method and application thereof
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Paragraph 0891-0892; 0893-0894, (2020/07/02)
The invention discloses a polycyclic compound, and a preparation method and an application thereof. The invention provides the polycyclic compound represented by formula I, or a pharmaceutically acceptable salt thereof. The compound has a relatively good inhibition effect on CDK7.
Further evidence for 2-alkyl-2-carboxyazetidines as γ-turn inducers
Baeza, Jose Luis,Gerona-Navarro, Guillermo,Thompson, Kevin,De Vega, M. Jesus Perez,Infantes, Lourdes,Garcia-Lopez, M. Teresa,Gonzalez-Muniz, Rosario,Martin-Martinez, Mercedes
supporting information; experimental part, p. 8203 - 8211 (2010/02/17)
(Chemical Equation Presented) Reverse turns, a common motif in proteins and peptides, have attracted attention due to their relevance in a wide variety of biological processes. In an attempt to artificially imitate and stabilize these turns in short pepti