Control of parasites in animals by the use of novel trifluoromethanesulfonanilide oxime ether derivatives
Novel trifluoromethanesulfonanilide oxime ether compounds useful for controlling endo and/or ectoparasites in the environment are provided, together with methods of making the same, and methods of using the inventive compounds to treat parasite infestations in vivo or ex vivo.
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Page/Page column 29
(2010/10/20)
1-Benzyloxy-4,5-dihydro-1H-imidazol-2-yl-amines, a novel class of NR1/2B subtype selective NMDA receptor antagonists
Screening of the Roche compound depository led to the identification of (1-benzyloxy-4,5-dihydro-1H-imidazol-2-yl)-butyl amine 4, a structurally novel NR1/2B subtype selective NMDA receptor antagonist. The structure-activity relationships developed in this series resulted in the discovery of a novel class of potent and selective NMDA receptor blockers displaying activity in vivo.
Synthesis of 1,2-oxazaheterocycles containing an isoindolone moiety from N-hydroxyphthalimide
Syntheses of the isoindolobenzoxazinone 1a and thienoxazinoisoindolones 1b,c was developed from N-hydroxyphthalimide 3 and halogenomethylaryl derivatives. The resulting aryloxy phthalimides 4a-c were reduced to hydroxylactams 5a-c which cyclized in acidic
Bartovic,Decroix,Netchitailo
p. 827 - 830
(2007/10/03)
Phosphoramidates and thiophosphoramidates as pesticides
Compounds of the formula STR1 and X is hydrogen, halo, alkyl, cyano or nitro, Y is oxygen or sulfur and R is lower alkyl, have been found to be excellent pesticides.
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(2008/06/13)
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