548453-22-1Relevant articles and documents
Synthesis, molecular docking, and QSAR study of bis-sulfonamide derivatives as potential aromatase inhibitors
Leechaisit, Ronnakorn,Pingaew, Ratchanok,Prachayasittikul, Veda,Worachartcheewan, Apilak,Prachayasittikul, Supaluk,Ruchirawat, Somsak,Prachayasittikul, Virapong
, (2019/08/14)
A library of bis-sulfonamides (9–26) were synthesized and tested for their aromatase inhibitory activities. Interestingly, all bis-sulfonamide derivatives inhibited the aromatase with IC50 range of 0.05–11.6 μM except for compound 23. The analo
Disulfonyl aryl diamine urease inhibitors as well as preparation method and application thereof
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Paragraph 0037-0040; 0042, (2019/01/14)
Disulfonyl aryl diamine compounds have the general structural formula shown in the description. The compounds have better inhibition functions on urease and can be used for preparing drugs for resisting gastritis, gastric ulcer, lithangiuria and the like.