Oxaziridine-mediated amination of primary amines: Scope and application to a one-pot pyrazole synthesis
(Chemical Equation Presented) Electrophilic amination of primary aliphatic and aromatic amines is reported using a diethylketomalonate-derived oxaziridine to afford the corresponding N-Boc hydrazines in good to excellent yields. The method allows a one-pot synthesis of pyrazoles from primary amines.
Armstrong, Alan,Jones, Lyn H.,Knight, Jamie D.,Kelsey, Richard D.
p. 713 - 716
(2007/10/03)
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