- Application of new cryptolepine derivatives in controlling and preventing plant-derived germs
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The invention relates to the technical field of natural medicinal chemistry and biopesticide, and discloses application of any one compound of 1a-24a of new cryptolepine derivatives in the preparationof a medicament for controlling or resisting rice blast
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Paragraph 0013-0017; 0032-0034
(2019/01/14)
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- Fluoroquinolones from imidoylketenes and iminopropadienones, RN≤C≤C≤C≤O
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3-Fluoro-, 4-fluoro-, and 2,3,4-trifluorophenyliminopropadienones have been generated by flash vacuum thermolysis (FVT) of 5-[(fluoroarylamino) methoxymethylene]-2,2-dimethyldioxan-4,6-dione (Meldrum's acid) derivatives. Their reaction with methanol affor
- Fulloon, Belinda E.,Wentrup, Curt
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experimental part
p. 115 - 120
(2009/08/15)
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- 3-GUANIDINOCARBONYL-1-HETEROARYL-INDOLE DERIVATIVES, PREPARATION PROCESS, THEIR USE AS MEDICAMENTS, AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM
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The present invention relates to 3-guanidinocarbonyl-1-heteroaryl-indole derivatives of the formula (I) in which R1 to R5 and Ar have the meaning stated in the claims. The inventive compounds are suitable for example as antiarrhytmic medicaments with cardioprotective component for infarction prophylaxis and infarction treatment and for the treatment of angina pectoris. They also inhibit in a preventive manner the pathophysiological processes associated with the development of ischemia-induced damage, in particular in the triggering of ischemia-induced cardiac arrhytmias and of heart failure.
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