681283-10-3Relevant articles and documents
Indium-Mediated Atom-Transfer and Reductive Radical Cyclizations of Iodoalkynes: Synthesis and Biological Evaluation of HIV-Protease Inhibitors
Yanada, Reiko,Koh, Yasuhiro,Nishimori, Nobuaki,Matsumura, Akira,Obika, Shingo,Mitsuya, Hiroaki,Fujii, Nobutaka,Takemoto, Yoshiji
, p. 2417 - 2422 (2007/10/03)
Novel indium-mediated radical cyclization reactions of aliphatic iodoalkynes have been studied. Treatment of iodoalkynes with a catalytic amount of In (0.1 equiv) and I2 (0.05 equiv) promotes atom-transfer 5-exo cyclization to give five-membere