Design, synthesis and structure-activity relationship of novel RXR-selective modulators
The synthesis and in vitro characterization of novel RXR-selective ligands possessing various substituted 1-benzofuran or 1-benzothiophene moieties are described.
Michellys, Pierre-Yves,D'Arrigo, Jennifer,Grese, Timothy A.,Karanewsky, Donald S.,Leibowitz, Mark D.,Mais, Dale A.,Mapes, Christopher M.,Reifel-Miller, Anne,Rungta, Deepa,Boehm, Marcus F.