Synthesis of a 1,3,5-benzotriazepine-2,4-dione based library
A library of benzotriazepines have been synthesised employing microwave-mediated synthesis, supported resins and parallel synthesis methodology.
Chuckowree, Irina,Ali Syed, Murtaza,Getti, Giulia,Parbhu Patel, Asha,Garner, Hannah,Tizzard, Graham J.,Coles, Simon J.,Spencer, John
supporting information; experimental part
p. 3607 - 3611
(2012/09/11)
Achiral, selective CCK2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template
Novel, achiral 1H-1,3,5-benzotriazepine-2,4(3H,5H)-diones have been prepared and structurally characterized. These compounds are potent CCK2 receptor antagonists that display a high degree of selectivity over CCK1 receptors.
Spencer, John,Gaffen, John,Griffin, Eric,Harper, Elaine A.,Linney, Ian D.,McDonald, Iain M.,Roberts, Sonia P.,Shaxted, Mark E.,Adatia, Trushar,Bashall, Alan
p. 2974 - 2983
(2008/09/19)
BENZOTRIAZEPINE DERIVATIVES AND THEIR USE AS GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS
This invention relates to a compound of formula (I). The compound is useful for the treatment of gastrin related disorders.
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Page/Page column 30
(2010/02/09)
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