- Synthesis of irreversibly binding bicalutamide analogs for imaging studies
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A new synthetic methodology for preparing radioactive androgen receptor binding compounds in order to determine receptor-ligands interactions has been developed.
- Nair, Vipin A.,Mustafa, Suni M.,Mohler, Michael L.,Yang, Jun,Kirkovsky, Leonid I.,Dalton, James T.,Miller, Duane D.
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p. 4821 - 4823
(2007/10/03)
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- Haloacetamide and azide substituted compounds and methods of use thereof
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The present invention relates to a novel class of anti-cancer compounds, which contain a haloacetamide or azide moiety and are, in one embodiment, alkylating agents. These agents, either alone or in a composition, are useful for treating cancer, preventin
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- HALOACETAMIDE AND AZIDE SUBSTITUTED COMPOUNDS AND METHODS OF USE THEREOF
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The present invention relates to a novel class of anti-cancer compounds, which contain a haloacetamide or azide moiety and are, in one embodiment, alkylating agents. These agents, either alone or in a composition, are useful for treating cancer, preventin
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Page/Page column 121-122; 130
(2008/06/13)
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- Synthesis of novel iodo derived bicalutamide analogs
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A series of optically active nonsteroidal selective androgen receptor modulators with structures analogous to bicalutamide was prepared by replacing the trifluoromethyl group with iodine and the sulfonyl linker by oxygen.
- Nair, Vipin A.,Mustafa, Suni M.,Mohler, Michael L.,Fisher, Scott J.,Dalton, James T.,Miller, Duane D.
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p. 9475 - 9477
(2007/10/03)
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