Synthesis and antiprotozoal activities of benzyl phenyl ether diamidine derivatives
Sixty-two cationic benzyl phenyl ether derivatives (36 amidines and 26 prodrugs) were prepared and assayed for activities in vitro and in vivo against Trypanosoma brucei rhodesiense (STIB900), and in vitro against Plasmodium falciparum (K1) and Leishmania
Patrick, Donald A.,Bakunov, Stanislav A.,Bakunova, Svetlana M.,Jones, Susan Kilgore,Wenzler, Tanja,Barszcz, Todd,Kumar, Arvind,Boykin, David W.,Werbovetz, Karl A.,Brun, Reto,Tidwell, Richard R.
p. 310 - 324
(2013/10/01)
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