1002557-03-0Relevant articles and documents
STAT DEGRADERS AND USES THEREOF
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Paragraph 001006; 001007, (2021/09/26)
The present invention provides compounds, compositions thereof, and methods of using the same.
Optimization of triarylimidazoles for Tie2: Influence of conformation on potency
Johnson, Neil W.,Semones, Marcus,Adams, Jerry L.,Hansbury, Michael,Winkler, Jim
, p. 5514 - 5517 (2008/03/11)
In an effort to understand the effect of N-alkylation of triarylimidazoles on Tie2 inhibition, ortho-substituted C-2 aryl analogs were synthesized to investigate the effect of different torsion angles on potency. This exercise resulted in the identificati