100304-64-1Relevant articles and documents
Opioid Agonists an Antagonists. Peptides Containing N-Terminal Allyl Groups and/or a Thiomethylene Linkage in Place of a Peptide Bond
Balboni, Gianfranco,Salvadori, Severo,Marastoni, Mauro,Tomatis, Roberto,Borea, Pier A.,Bianchi, Clementina
, p. 1645 - 1652 (2007/10/02)
Peptides containing N-allyl or N,N-diallyl groups at the N-terminus have been synthesized as potential opioid antagonists.A number of analogues with an amine bond replaced by a thiomethylene group have also been prepared.In brain binding assays and in gui