1067228-95-8Relevant articles and documents
2-Aryl-3,6-dialkyl-5-dialkylaminopyrimidin-4-ones as novel CRF-1 receptor antagonists
Hodgetts, Kevin J.,Yoon, Taeyoung,Huang, Jianhua,Gulianello, Michael,Kieltyka, Andrzej,Primus, Renee,Brodbeck, Robbin,De Lombaert, Stephane,Doller, Dario
, p. 2497 - 2500 (2003)
The discovery, synthesis and structure-activity studies of a novel series of 2-arylpyrimidin-4-ones as CRF-1 receptor antagonists is described. These compounds are structurally simple and display appropriate physical properties for CNS agents