Nucleosides, nucleotides and nucleic acids p. 1797 - 1811 (2004)
Update date:2022-08-11
Topics:
Wu
Xiao
Jiang
Fu
Ju
Zhao
A series of N-diisopropylphosphoryl (DIPP) L-amino acid ester prodrugs of zidovudine (AZT) (3a-3e) and stavudine (d4T) (4a-4e) has been prepared. The activity of these compounds against MCF-7 cells (human pleural effusion breast adenocarcinoma cell line)
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