Bioorganic and Medicinal Chemistry Letters p. 4045 - 4050 (2004)
Update date:2022-08-16
Topics:
Bauer, Shawn M.
Goldman, Erick A.
Huang, Wenrong
Su, Ting
Wang, Lingyan
Woolfrey, John
Wu, Yanhong
Zuckett, Jingmei F.
Arfsten, Ann
Huang, Brian
Kothule, Jaya
Lin, Joyce
May, Bridget
Sinha, Uma
Wong, Paul W.
Hutchaleelaha, Athiwat
Scarborough, Robert M.
Zhu, Bing-Yan
Parallel synthesis and iterative optimization led to the discovery of a series of potent and specific factor Xa inhibitors demonstrating excellent in vitro activity with promising pharmacokinetics.
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(2004)