Aromatic and amine substituent effects on the apparent lipophilicities of N-[(2-pyrrolidinyl)methyl]-substituted benzamides

DOI: 10.1002/jps.2600830309

Source and publish data:

Journal of Pharmaceutical Sciences p. 305 - 315 (1994)

Update date:2022-08-29

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Authors:

Schmidt Schmidt

Votaw Votaw

Kessler Kessler

De Paulis

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Article abstract of DOI:10.1002/jps.2600830309

Lipophilic properties of 92 dopamine D-2 receptor antagonists belonging to the substituted benzamide class of compounds (orthopramides and methoxysalicylamides) were determined by octadecylsilane reversed-phase HPLC. The apparent lipophilicity at pH 7.5 (

Full text of DOI:10.1002/jps.2600830309

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