European Journal of Medicinal Chemistry p. 193 - 210 (2018)
Update date:2022-08-15
Topics:
Reddy, Damodara N.
Singh, Sukrit
Ho, Chris M.W.
Patel, Janki
Schlesinger, Paul
Rodgers, Stephen
Doctor, Allan
Marshall, Garland R.
Gramicidin A, a topical antibiotic made from alternating L and D amino acids, is characterized by its wide central pore; upon insertion into membranes, it forms channels that disrupts ion gradients. We present helical peptidomimetics with this characteris
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