1-(1-Benzylaziridine-2-sulfonyl)pyrrolidine

Base Information

Chemical Name:1-(1-Benzylaziridine-2-sulfonyl)pyrrolidine
CAS No.:87975-48-2
Molecular Formula:C₁₃H₁₈N₂O₂S
Molecular Weight:266.364
Hs Code.:
DSSTox Substance ID:DTXSID40579427

Synonyms:1-(1-Benzylaziridine-2-sulfonyl)pyrrolidine;87975-48-2;DTXSID40579427;AKOS015907514;1-(1-benzylaziridin-2-yl)sulfonylpyrrolidine;1-[(1-benzyl-2-aziridinyl)sulfonyl]pyrrolidine

Suppliers and Price of 1-(1-Benzylaziridine-2-sulfonyl)pyrrolidine

Supply Marketing:

Business phase:: The product has achieved commercial mass production^*data from LookChem market partment

Manufacturers and distributors:

Manufacture/Brand
Chemicals and raw materials
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price

Total 1 raw suppliers

Chemical Property of 1-(1-Benzylaziridine-2-sulfonyl)pyrrolidine

Chemical Property:

XLogP3:1.5
Hydrogen Bond Donor Count:0
Hydrogen Bond Acceptor Count:4
Rotatable Bond Count:4
Exact Mass:266.10889899
Heavy Atom Count:18
Complexity:378

Purity/Quality:: 99% ^*data from raw suppliers

Safty Information:

Pictogram(s):
Hazard Codes:

MSDS Files:: SDS file from LookChem

Useful:

Canonical SMILES:C1CCN(C1)S(=O)(=O)C2CN2CC3=CC=CC=C3

Technology Process of 1-(1-Benzylaziridine-2-sulfonyl)pyrrolidine

There total 6 articles about 1-(1-Benzylaziridine-2-sulfonyl)pyrrolidine which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield:

: 87975-23-3
Benzyl-[2-bromo-2-(pyrrolidine-1-sulfonyl)-ethyl]-amine

: 87975-48-2
1-(1-Benzyl-aziridine-2-sulfonyl)-pyrrolidine

Guidance literature:: With triethylamine; In dimethyl sulfoxide; at 75 ℃; for 4h; Yield given;
DOI:10.1055/s-1983-30527

Reference yield:

: 87975-58-4
vinyl sulfonamide of pyrrolidine

: 87975-48-2
1-(1-Benzyl-aziridine-2-sulfonyl)-pyrrolidine

Guidance literature:: Multi-step reaction with 3 steps

1: 83 percent / Br₂ / CCl₄ / 48 h / Ambient temperature

2: 80 percent / triethylamine / benzene / 24 h / Ambient temperature

3: dimethylsulfoxide / 4 h / 75 °C

With bromine; triethylamine; In tetrachloromethane; dimethyl sulfoxide; benzene;
DOI:10.1055/s-1983-30527

Reference yield:

: 87975-60-8
1-(1,2-Dibromo-ethanesulfonyl)-pyrrolidine

: 87975-48-2
1-(1-Benzyl-aziridine-2-sulfonyl)-pyrrolidine

Guidance literature:: Multi-step reaction with 2 steps

1: 80 percent / triethylamine / benzene / 24 h / Ambient temperature

2: dimethylsulfoxide / 4 h / 75 °C

With triethylamine; In dimethyl sulfoxide; benzene;
DOI:10.1055/s-1983-30527