4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenylboronic acid

Base Information

• Chemical Name: 4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenylboronic acid
• CAS No.: 943742-47-0
• Molecular Formula: C₂₃H₂₃BN₂O₆
• Molecular Weight: 434.256

Synonyms:4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenylboronic acid

Chemical Property of 4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenylboronic acid

Chemical Property:

Purity/Quality:

Safty Information:

• Pictogram(s):  
• Hazard Codes: 

MSDS Files:

Useful:

Technology Process of 4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenylboronic acid

There total 1 articles about 4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenylboronic acid which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield: 72.0%

{3-[2-(4-bromo-phenoxy)-acetylamino]-benzyl}-carbamic acid benzyl ester (943742-46-9) + 2-(5,5-dimethyl-1,3,2-dioxaborinan-2-yl)-5,5-dimethyl-1,3,2-dioxaborinane (201733-56-4) → 4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenylboronic acid (943742-47-0)

Guidance literature:

With potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride; In dimethyl sulfoxide; at 80 ℃; for 3h;

Reference yield: 68.0%

imidodicarbonic acid 2-(6-amino-1-isoquinolinyl)-1,3-bis(1,1-dimethylethyl)ester (745020-22-8) + 4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenylboronic acid (943742-47-0) + Glyoxilic acid (298-12-4) → 2-(4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenyl)-2-(1-(bis(tert-butoxycarbonyl)amino)isoquinolin-6-ylamino)acetic acid (943742-48-1)

Guidance literature:

In N,N-dimethyl-formamide; acetonitrile; at 65 ℃; for 16h;

upstream raw materials:

{3-[2-(4-bromo-phenoxy)-acetylamino]-benzyl}-carbamic acid benzyl ester

2-(5,5-dimethyl-1,3,2-dioxaborinan-2-yl)-5,5-dimethyl-1,3,2-dioxaborinane

Downstream raw materials:

2-(4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenyl)-2-(1-(bis(tert-butoxycarbonyl)amino)isoquinolin-6-ylamino)acetic acid

Post a RFQ

Cas No.:

Product Name:

Quantity:

Please select Metric Ton KG G Pound L ML

Email:

Company name:

Valid Period:

Detailed Requirements:

• Sample
• MOQ
• GMP
• FDA
• Price
  FOB CIF CFR EXW
• Urgent purchase

Enter 15 to 2000 letters.Word count: 0 letters

Attach files(File Format: Jpeg, Jpg, Gif, Png, PDF, PPT, Zip, Rar,Word or Excel Maximum File Size: 3MB)

Remove

Submit

1

What can I do for you?
Get Best Price

Get Best Price for 943742-47-0 4-(2-(3-((benzyloxycarbonylamino)methyl)phenylamino)-2-oxoethoxy)phenylboronic acid

Send

Send

Metric Ton KG G Pound L ML

Send

Send