{[(2S,3S)-3-ethynyl-3-methyl-1-(toluene-4-sulfonyl)-aziridine-2-carbonyl]amino}acetic acid methyl ester

Base Information

• Chemical Name: {[(2S,3S)-3-ethynyl-3-methyl-1-(toluene-4-sulfonyl)-aziridine-2-carbonyl]amino}acetic acid methyl ester
• CAS No.: 916346-74-2
• Molecular Formula: C₁₆H₁₈N₂O₅S
• Molecular Weight: 350.395

Synonyms:{[(2S,3S)-3-ethynyl-3-methyl-1-(toluene-4-sulfonyl)-aziridine-2-carbonyl]amino}acetic acid methyl ester

Chemical Property of {[(2S,3S)-3-ethynyl-3-methyl-1-(toluene-4-sulfonyl)-aziridine-2-carbonyl]amino}acetic acid methyl ester

Chemical Property:

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Technology Process of {[(2S,3S)-3-ethynyl-3-methyl-1-(toluene-4-sulfonyl)-aziridine-2-carbonyl]amino}acetic acid methyl ester

There total 1 articles about {[(2S,3S)-3-ethynyl-3-methyl-1-(toluene-4-sulfonyl)-aziridine-2-carbonyl]amino}acetic acid methyl ester which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield: 100.0%

C16H20N2O6S (960595-70-4) → {[(2S,3S)-3-ethynyl-3-methyl-1-(toluene-4-sulfonyl)-aziridine-2-carbonyl]amino}acetic acid methyl ester (916346-74-2)

Guidance literature:

With triphenylphosphine; diethylazodicarboxylate;

DOI:10.1021/ja0758077

Reference yield: 60.0%

{[(2S,3S)-3-ethynyl-3-methyl-1-(toluene-4-sulfonyl)-aziridine-2-carbonyl]amino}acetic acid methyl ester (916346-74-2) + isovanillin (621-59-0) → [(2S,3R)-3-(5-formyl-2-methoxyphenoxy)-3-methyl-2-(toluene-4-sulfonylamino)pent-4-ynoylamino]acetic acid methyl ester

Guidance literature:

With copper (I) acetate; 1,8-diazabicyclo[5.4.0]undec-7-ene; In toluene; at 20 ℃; for 2h;

DOI:10.1021/ol062010w

Reference yield: 42.0%

{[(2S,3S)-3-ethynyl-3-methyl-1-(toluene-4-sulfonyl)-aziridine-2-carbonyl]amino}acetic acid methyl ester (916346-74-2) + p-cresol (106-44-5) → [(2S,3R)-3-methyl-2-(toluene-4-sulfonylamino)-3-p-tolyloxypent-4-ynoylamino]acetic acid methyl ester

Guidance literature:

With copper (I) acetate; 1,8-diazabicyclo[5.4.0]undec-7-ene; In toluene; at 20 ℃;

DOI:10.1021/ol062010w DOI:10.1021/ja0758077

upstream raw materials:

C₁₆H₂₀N₂O₆S

Downstream raw materials:

C₃₅H₃₇N₃O₁₁S

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