Technology Process of C17H18ClIN4O3
There total 3 articles about C17H18ClIN4O3 which
guide to synthetic route it.
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synthetic route:
- Guidance literature:
-
With
1-hydroxy-7-aza-benzotriazole; N-ethyl-N,N-diisopropylamine; HATU;
In
N,N-dimethyl-formamide;
at 80 ℃;
DOI:10.1016/j.bmcl.2012.12.014
- Guidance literature:
-
Multi-step reaction with 2 steps
1: trifluoroacetic acid / dichloromethane / 20 °C
2: N-ethyl-N,N-diisopropylamine; HATU; 1-hydroxy-7-aza-benzotriazole / N,N-dimethyl-formamide / 80 °C
With
1-hydroxy-7-aza-benzotriazole; N-ethyl-N,N-diisopropylamine; HATU; trifluoroacetic acid;
In
dichloromethane; N,N-dimethyl-formamide;
DOI:10.1016/j.bmcl.2012.12.014
- Guidance literature:
-
Multi-step reaction with 3 steps
1: caesium carbonate / N,N-dimethyl-formamide / 0 - 20 °C
2: trifluoroacetic acid / dichloromethane / 20 °C
3: N-ethyl-N,N-diisopropylamine; HATU; 1-hydroxy-7-aza-benzotriazole / N,N-dimethyl-formamide / 80 °C
With
1-hydroxy-7-aza-benzotriazole; caesium carbonate; N-ethyl-N,N-diisopropylamine; HATU; trifluoroacetic acid;
In
dichloromethane; N,N-dimethyl-formamide;
DOI:10.1016/j.bmcl.2012.12.014