2-(4-phenyl-[1,2,3]triazol-1-yl)-1S-(2-thiophen-2-yl-acetylamino)ethaneboronic acid

Base Information

Chemical Name:2-(4-phenyl-[1,2,3]triazol-1-yl)-1S-(2-thiophen-2-yl-acetylamino)ethaneboronic acid
CAS No.:1429666-57-8
Molecular Formula:C₁₆H₁₇BN₄O₃S
Molecular Weight:356.213
Hs Code.:

Synonyms:2-(4-phenyl-[1,2,3]triazol-1-yl)-1S-(2-thiophen-2-yl-acetylamino)ethaneboronic acid

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Chemical Property of 2-(4-phenyl-[1,2,3]triazol-1-yl)-1S-(2-thiophen-2-yl-acetylamino)ethaneboronic acid

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Technology Process of 2-(4-phenyl-[1,2,3]triazol-1-yl)-1S-(2-thiophen-2-yl-acetylamino)ethaneboronic acid

There total 2 articles about 2-(4-phenyl-[1,2,3]triazol-1-yl)-1S-(2-thiophen-2-yl-acetylamino)ethaneboronic acid which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield: 85.0%

: 1429666-52-3
(+)-pinanediol 2-(4-phenyl-[1,2,3]triazol-1-yl)-1S-(2-thiophen-2-yl-acetylamino)ethaneboronate ester

: 1429666-57-8
2-(4-phenyl-[1,2,3]triazol-1-yl)-1S-(2-thiophen-2-yl-acetylamino)ethaneboronic acid

Guidance literature:: With hydrogenchloride; water; phenylboronic acid; In hexane; acetonitrile; Inert atmosphere;

Reference yield:

: 1425968-44-0
(+)-pinanediol (1R)-2-azido-1-[(2-thienylacetyl)amino]ethaneboronate

: 1429666-57-8
2-(4-phenyl-[1,2,3]triazol-1-yl)-1S-(2-thiophen-2-yl-acetylamino)ethaneboronic acid

Guidance literature:: Multi-step reaction with 2 steps

1: sodium L-ascorbate; copper(II) sulfate / tert-butyl alcohol; water / 2 h / 60 °C / Inert atmosphere; Sealed tube

2: phenylboronic acid; hydrogenchloride / hexane; water; acetonitrile / Inert atmosphere

With hydrogenchloride; copper(II) sulfate; sodium L-ascorbate; phenylboronic acid; In hexane; water; acetonitrile; tert-butyl alcohol;
DOI:10.1021/acs.jmedchem.5b00341