[(4-amino-benzyl)-tert-butoxycarbonylmethylamino]acetic acid tert-butyl ester

Base Information

• Chemical Name: [(4-amino-benzyl)-tert-butoxycarbonylmethylamino]acetic acid tert-butyl ester
• CAS No.: 1088539-80-3
• Molecular Formula: C₁₉H₃₀N₂O₄
• Molecular Weight: 350.458

Synonyms:[(4-amino-benzyl)-tert-butoxycarbonylmethylamino]acetic acid tert-butyl ester

Chemical Property of [(4-amino-benzyl)-tert-butoxycarbonylmethylamino]acetic acid tert-butyl ester

Chemical Property:

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Technology Process of [(4-amino-benzyl)-tert-butoxycarbonylmethylamino]acetic acid tert-butyl ester

There total 1 articles about [(4-amino-benzyl)-tert-butoxycarbonylmethylamino]acetic acid tert-butyl ester which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield: 59.0%

bromoacetic acid tert-butyl ester (5292-43-3) + (4-aminomethyl)aniline (4403-71-8) → [(4-amino-benzyl)-tert-butoxycarbonylmethylamino]acetic acid tert-butyl ester (1088539-80-3)

Guidance literature:

With potassium carbonate; potassium iodide; In acetonitrile; for 25h; Reflux;

DOI:10.1002/anie.200802242

Reference yield:

[(4-amino-benzyl)-tert-butoxycarbonylmethylamino]acetic acid tert-butyl ester (1088539-80-3) + 4,4'-(cyclopent-1-ene-1,2-diyl)bis(5-methylthiophene-2-carbonyl chloride) (331432-80-5) → C36H43ClN2O6S2

Guidance literature:

With triethylamine; In tetrahydrofuran; at 20 ℃; for 5.5h; Inert atmosphere;

DOI:10.1002/anie.200802242

Reference yield:

[(4-amino-benzyl)-tert-butoxycarbonylmethylamino]acetic acid tert-butyl ester (1088539-80-3) + 4,4'-(cyclopent-1-ene-1,2-diyl)bis(5-methylthiophene-2-carbonyl chloride) (331432-80-5) → {[4-({4-[2-(5-{4-[(bis-tert-butoxycarbonylmethylamino)methyl]phenylcarbamoyl}-2-methylthiophen-3-yl)cyclopent-1-enyl]-5-methylthiophene-2-carbonyl}amino)benzyl]tert-butoxycarbonylmethylamino}acetic acid tert-butyl ester (1088539-87-0)

Guidance literature:

With triethylamine; In tetrahydrofuran; Inert atmosphere;

DOI:10.1002/anie.200802242

upstream raw materials:

bromoacetic acid tert-butyl ester

(4-aminomethyl)aniline

Downstream raw materials:

{[4-({4-[2-(5-{4-[(bis-tert-butoxycarbonylmethylamino)methyl]phenylcarbamoyl}-2-methylthiophen-3-yl)cyclopent-1-enyl]-5-methylthiophene-2-carbonyl}amino)benzyl]tert-butoxycarbonylmethylamino}acetic acid tert-butyl ester

C₄₄H₇₀N₂O₅

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