(S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester

Base Information

Chemical Name:(S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester
CAS No.:463313-56-6
Molecular Formula:C₃₄H₄₃F₅N₂O₁₅
Molecular Weight:814.712
Hs Code.:

(S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester

Synonyms:

Suppliers and Price of (S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester

Supply Marketing:

Business phase:: The product has achieved commercial mass production^*data from LookChem market partment

Manufacturers and distributors:

Manufacture/Brand
Chemicals and raw materials
Packaging
price

Total 0 raw suppliers

Chemical Property of (S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester

Chemical Property:

Purity/Quality:

Safty Information:

Pictogram(s):
Hazard Codes:

MSDS Files:

Useful:

Technology Process of (S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester

There total 6 articles about (S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield:

: 7536-58-5,98482-77-0
BOC-L-aspartic acid 4-benzyl ester

: 463313-56-6
(S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester

Guidance literature:: Multi-step reaction with 4 steps

1: 93 percent / DCC / ethyl acetate / 1 h / 0 - 20 °C

2: 95 percent / ethyl acetate / 20 °C

3: H₂ / Pd/C / ethanol; acetic acid / 1 h / 25 °C / 750.06 Torr

4: DCC / ethyl acetate / 1 h / 0 - 20 °C

With hydrogen; dicyclohexyl-carbodiimide; palladium on activated charcoal; In ethanol; acetic acid; ethyl acetate;
DOI:10.1016/S0957-4166(02)00212-4

Reference yield:

: 82825-48-7
α-pentafluorophenyl N-tert-butoxycarbonyl-β-benzyl-L-asparaginate

: 463313-56-6
(S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester

Guidance literature:: Multi-step reaction with 3 steps

1: 95 percent / ethyl acetate / 20 °C

2: H₂ / Pd/C / ethanol; acetic acid / 1 h / 25 °C / 750.06 Torr

3: DCC / ethyl acetate / 1 h / 0 - 20 °C

With hydrogen; dicyclohexyl-carbodiimide; palladium on activated charcoal; In ethanol; acetic acid; ethyl acetate;
DOI:10.1016/S0957-4166(02)00212-4

Reference yield:

: 142825-49-8
5-<(benzyloxycarbonyl)amino>pentyl 2,3,4,6-tetra-O-acetyl-β-D-glucopyranoside

: 463313-56-6
(S)-3-tert-Butoxycarbonylamino-N-[5-((2R,3R,4S,5R,6R)-3,4,5-triacetoxy-6-acetoxymethyl-tetrahydro-pyran-2-yloxy)-pentyl]-succinamic acid pentafluorophenyl ester

Guidance literature:: Multi-step reaction with 4 steps

1: 96 percent / H₂ / Pd/C / ethanol; acetic acid / 1 h / 25 °C / 750.06 Torr

2: 95 percent / ethyl acetate / 20 °C

3: H₂ / Pd/C / ethanol; acetic acid / 1 h / 25 °C / 750.06 Torr

4: DCC / ethyl acetate / 1 h / 0 - 20 °C

With hydrogen; dicyclohexyl-carbodiimide; palladium on activated charcoal; In ethanol; acetic acid; ethyl acetate;
DOI:10.1016/S0957-4166(02)00212-4