(S)-2-{(S)-6-Benzyloxycarbonylamino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester

Base Information

• Chemical Name: (S)-2-{(S)-6-Benzyloxycarbonylamino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester
• CAS No.: 161147-15-5
• Molecular Formula: C₅₂H₆₃N₅O₁₀
• Molecular Weight: 918.1

Synonyms:

Chemical Property of (S)-2-{(S)-6-Benzyloxycarbonylamino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester

Chemical Property:

Purity/Quality:

Safty Information:

• Pictogram(s):  
• Hazard Codes: 

MSDS Files:

Useful:

Technology Process of (S)-2-{(S)-6-Benzyloxycarbonylamino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester

There total 1 articles about (S)-2-{(S)-6-Benzyloxycarbonylamino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester which guide to synthetic route it. The literature collected by LookChem mainly comes from the sharing of users and the free literature resources found by Internet computing technology. We keep the original model of the professional version of literature to make it easier and faster for users to retrieve and use. At the same time, we analyze and calculate the most feasible synthesis route with the highest yield for your reference as below:

synthetic route:

Reference yield:

2,5-dioxopyrrolidin-1-yl N-(tert-butoxycarbonyl)-L-tryptophanate (3392-11-8) + (S)-2-((S)-2-Amino-6-benzyloxycarbonylamino-hexanoylamino)-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester; compound with trifluoro-acetic acid → (S)-2-{(S)-6-Benzyloxycarbonylamino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester (161147-15-5)

Guidance literature:

With benzotriazol-1-ol; N-ethyl-N,N-diisopropylamine; In N,N-dimethyl-formamide; for 24h; Yield given; Ambient temperature;

DOI:10.1135/cccc19942511

Reference yield:

(S)-2-{(S)-6-Benzyloxycarbonylamino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester (161147-15-5) → (S)-2-{(S)-6-Amino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester

Guidance literature:

With hydrogen; palladium on activated charcoal; In methanol; for 6.5h; Ambient temperature;

DOI:10.1135/cccc19942511

Reference yield:

(S)-2-{(S)-6-Benzyloxycarbonylamino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester (161147-15-5) → (S)-2-[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-6-(3-phenyl-ureido)-hexanoylamino]-succinic acid 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester

Guidance literature:

Multi-step reaction with 2 steps

1: H₂ / Pd-C / methanol / 6.5 h / Ambient temperature

2: N-ethyldiisopropylamine / dimethylformamide / 20 h / Ambient temperature

With hydrogen; N-ethyl-N,N-diisopropylamine; palladium on activated charcoal; In methanol; N,N-dimethyl-formamide;

DOI:10.1135/cccc19942511

upstream raw materials:

2,5-dioxopyrrolidin-1-yl N-(tert-butoxycarbonyl)-L-tryptophanate

Post a RFQ

Cas No.:

Product Name:

Quantity:

Please select Metric Ton KG G Pound L ML

Email:

Company name:

Valid Period:

Detailed Requirements:

• Sample
• MOQ
• GMP
• FDA
• Price
  FOB CIF CFR EXW
• Urgent purchase

Enter 15 to 2000 letters.Word count: 0 letters

Attach files(File Format: Jpeg, Jpg, Gif, Png, PDF, PPT, Zip, Rar,Word or Excel Maximum File Size: 3MB)

Remove

Submit

1

What can I do for you?
Get Best Price

Get Best Price for 161147-15-5 (S)-2-{(S)-6-Benzyloxycarbonylamino-2-[(S)-2-tert-butoxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-hexanoylamino}-succinic acid 4-benzyl ester 1-[2-(2,4,6-trimethyl-phenyl)-ethyl] ester

Send

Send

Metric Ton KG G Pound L ML

Send

Send