14465-74-8Relevant articles and documents
Regioselective synthesis of annulated quinoline and pyridine derivatives by silver-catalyzed 6-endo-dig cycloisomerization
Majumdar,Nandi, Raj Kumar,Ganai, Sintu,Taher, Abu
, p. 116 - 120 (2011)
3H-pyrano[3,2-f]quinoline-3-one, 4-methyl-4,7-phen-anthrolin-3(4H)-one, and 1,3-dimethylpyrido[3,2-d]pyrimidine-2,4(1H,3H)-dione derivatives have been synthesized by hitherto unreported silver-catalyzed 6-endo-dig mode of cycloisomerization from various N-propargylated heterocyclic compounds. The silver-catalyzed reaction provides the synthesis of potential bioactive compounds in excellent yields. Georg Thieme Verlag Stuttgart - New York.
(3-(1H-1,2,3-triazole)phenyl)phosphoric acid derivative as well as preparation method and application thereof
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Paragraph 0152, (2021/08/07)
The invention relates to the technical field of medicinal chemistry, and discloses a (3-(1H-1,2,3-triazole)phenyl)phosphoric acid derivative derivative as shown in a formula X which is described in the specification. The derivative has good and broad-spec
K2S2O8-Mediated Synthesis of Highly Functionalized Pyrroles via Oxidative Self-Dimerization of N-Propargylamines
Behera, Bipin Kumar,Sahu, Archana Kumari,Devi, Ngangbam Renubala,Saikia, Anil K.
, p. 12481 - 12493 (2021/09/20)
An efficient methodology has been developed for the synthesis of tetra- and pentasubstituted pyrroles via oxidative self-dimerization of N-propargylamines catalyzed by silver benzoate in the presence of K2S2O8 in good yields. The protocol provides a simple route for the synthesis of both tetra- and pentasubstituted pyrroles with two carbonyl groups in the side chain. The methodology can be extended toward the synthesis of pyrrolo[3,4-d]pyridazine.
Synthesis and biological evaluation of coumarin-linked 4-anilinomethyl-1,2,3-triazoles as potent inhibitors of carbonic anhydrases ix and xiii involved in tumorigenesis
Thacker, Pavitra S.,Tiwari, Prerna L.,Angeli, Andrea,Srikanth, Danaboina,Swain, Baijayantimala,Arifuddin, Mohammed,Supuran, Claudiu T.
, (2021/04/22)
A series of coumarin-linked 4-anilinomethyl-1,2,3-triazoles (6a–t) was synthesized via a molecular hybridization approach, through carbon C-6 of the coumarin moiety. The synthesized compounds were evaluated for their inhibition of carbonic anhydrase (CA)
