151860-16-1Relevant articles and documents
Synthesis of azabicyclo[3.1.0]amine analogues of anacardic acid as potent antibacterial agents
Vempati, Ravi Kumar,Reddy,Alapati, Srinivasa Rao,Dubey
, p. 986 - 994 (2013/06/26)
Azabicyclo[3.1.0]amine analogues of anacardic acid (16a, 16b, 18a, 18b, 19 and 19b) were synthesized from anacardic acid and tested for their antibacterial activity against Gram positive and Gram negative bacteria. Most of the compounds are having potency at par with ampicillin and inferior with other standard drugs.
Synthesis of an amino moiety in trovafloxacin by using an in-expensive amidine base, N, N-diethylacetamidine
Madhusudhan,Balraju,Rajesh,Narayana, B. Venkata,Reddy
experimental part, p. 569 - 573 (2009/12/06)
The simple and in-expensive amidine base, N.N-diethylacetamidine, has been prepared and utilized in the construction of bicyclic hetero compound, 4 and employed for further reduction of amidic carbonyl groups of 4 by using NaBH 4I2-THF condition which is an efficient and commercially viable method to prepare 5 towards the synthesis of amino moiety I, in Trovafloxacin 2 an antibacterial agent.
Process for preparing trovafloxacin acid salts
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Page column 12-13, (2008/06/13)
Trovafloxacin acid salts are prepared via the hydrolysis of imine intermediates using mineral acid including, but not limited to, methanesulfonic acid, ethanesulfonic acid, benzenesulfonic acid, nitric acid, sulfuric acid, phosphoric acid, hydrochloric ac