1004994-35-7Relevant academic research and scientific papers
Two-step N-acylindazole to N-alkylindazole reduction. Further synthetic studies on the serotonergic agonist AL-34662
Conrow, Raymond E.,Delgado, Pete,Dean, W. Dennis,Callen, Gary R.,Plummer, Scott V.
, p. 2348 - 2350 (2008/09/18)
A synthesis of the title compound, operable on kilogram scale, employs reductive acetylation of an N-acylindazole to give a hemiaminal acetate followed by deacetoxylation to the corresponding N-alkylindazole.
INTERMEDIATES AND METHODS FOR SEROTONERGIC AGONIST SYNTHESIS
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Page/Page column 3, (2010/11/29)
Disclosed is a method of making a 1-alkylindazole comprising reacting a 1-acylindazole with a first reducing agent, and contacting the resulting mixture with an acid anhydride or acyl halide, and with pyridine or a 4-dialkylaminopyridine or a combination
