1005161-95-4Relevant academic research and scientific papers
6-endo-dig Cyclization of heteroarylesters to alkynes promoted by Lewis acid catalyst in the presence of Br?nsted acid
Hellal, Malik,Bourguignon, Jean-Jacques,Bihel, Frédéric J.-J.
, p. 62 - 65 (2008/09/17)
We report a regiocontrolled 6-endo-dig cyclization of 2-(2-arylethynyl)heteroaryl esters occurred under Br?nsted acidic conditions and in the presence of a catalytic amount of Lewis acids such as Cu(OTf)2, AuCl3, or (CF3CO
