101817-00-9Relevant articles and documents
Synthesis of Cyclic and Cyclically Branched Tachykinine Partial Sequences. Part 3: Synthesis of the cyclo and of Two Ring-Expanded Analogues
Neubert, K.,Hartrodt, Bianka,Berger, Edith,Mehlis, B.,Rueger, Margitta,et al.
, p. 617 - 622 (2007/10/02)
The authors describe the synthesis of and of two analogues, the ring of which were expanded by the insertion of 1 or 2 molecules of ε-aminocaproic acid.The cyclopeptides had been tested for their activity as to the smooth musculature.The cyclo- as well as the analogue expanded by ε-aminocaproic acid exhibit a behaviour typically of the partial agonists.