102017-55-0Relevant academic research and scientific papers
Enantioselective Construction of Pyrimidine-Fused Diazepinone Derivatives Bearing a Tertiary Stereogenic Center Enabled by Iridium-Catalysed Intramolecular Allylic Substitution
Chan, Albert S. C.,Chan, Hoi Shan,Chen, Bin,He, Xiaobo,Jiang, Xiaoding,Liang, Hao,Pan, Bendu,Qian, Xu,Qiu, Liqin,Zhang, Yaqi
, p. 3227 - 3232 (2021/06/16)
The iridium-catalysed enantioselective intramolecular allylic substitution of pyrimidine-tethered allylic carbonates was developed. A wide range of chiral pyrimidine-fused diazepinone derivatives were successfully constructed in 88–96% yields with 85–99%
Synthesis of 2,4,5-trisubstituted pyrimidines
Pawar,Burungale,Karale
, p. 133 - 136 (2013/09/23)
A new series of 2,4,5-trisubstituted pyrimidines incorporating 1,3,4-thiadiazole and 1,2,4-triazole rings were synthesized and characterized by the spectral techniques.
