1022945-75-0Relevant articles and documents
Improvement in oral bioavailability of 2,4-diaminopyrimidine c-Met inhibitors by incorporation of a 3-amidobenzazepin-2-one group
Milkiewicz, Karen L.,Aimone, Lisa D.,Albom, Mark S.,Angeles, Thelma S.,Chang, Hong,Grobelny, Jennifer V.,Husten, Jean,LoSardo, Christine,Miknyoczki, Sheila,Murthy, Seetha,Rolon-Steele, Damaris,Underiner, Ted L.,Weinberg, Linda R.,Worrell, Candace S.,Zeigler, Kelli S.,Dorsey, Bruce D.
, p. 6274 - 6284 (2011/12/15)
The hepatocyte growth factor (HGF)-c-Met signaling axis is involved in the mediation of many biological activities, including angiogenesis, proliferation, cell survival, cell motility, and morphogenesis. Dysregulation of c-Met signaling (e.g., overexpress