1031337-85-5Relevant articles and documents
Imidazopyridines as VLA-4 integrin antagonists
Phillips, David J.,Davenport, Richard J.,Demaude, Thierry A.,Galleway, Fiona P.,Jones, Mark W.,Knerr, Laurent,Perry, Benjamin G.,Ratcliffe, Andrew J.
scheme or table, p. 4146 - 4149 (2009/04/07)
We describe a novel series of imidazopyridine substituted phenylalanines which are potent VLA-4 antagonists. A wide variety of substituents are tolerated as replacements for the pendant 3-pyridyl ring. A clear structure-activity relationship was identifie