103628-53-1Relevant articles and documents
Synthesis of carbon-14 labelled indolic 5HT1 receptor agonists
Waterhouse, Ian,Cable, Karl M.,Fellows, Ian,Wipperman, Mark D.,Sutherland, Derek R.
, p. 1021 - 1030 (2007/10/03)
Syntheses of carbon-14 labelled versions of indolic 5HT1 agonists sumatriptan (GR43175), GR40370 and naratriptan (GR85548) are described. Introduction of the label via cyanation of ketoformanilides, formed by oxidative cleavage of an indole rin
Indole derivative
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, (2008/06/13)
A compound of formula (I) STR1 and its physiologically acceptable salts and solvates are described as useful in treating and/or preventing pain resulting from dilatation of the cranial vasculature in particular migraine. The compound (I) may be prepared, for example, by cyclizing a compound of formula (II) STR2