104291-44-3Relevant articles and documents
Design, synthesis, and bioassay of 4-thiazolinone derivatives as influenza neuraminidase inhibitors
Xiao, Mengwu,Xu, Lvjie,Lin, Ding,Lian, Wenwen,Cui, Manying,Zhang, Meng,Yan, Xiaowei,Li, Shuishi,Zhao, Jun,Ye, Jiao,Liu, Ailin,Hu, Aixi
, (2021)
A series of 4-thiazolinone derivatives (D1-D58) were designed and synthesized. All of the derivatives were evaluated in vitro for neuraminidase (NA) inhibitory activities against influenza virus A (H1N1), and the inhibitory activities of the five most pot
A New, Convenient Synthesis of 1,6-Diaryl-2-thioxoperhydro-4-pyrimidinones: Reaction of 3-Phenyl-2-propenoyl Isothiocyanate With Aromatic and Heteroaromatic Amines
Hafez, Ebtisam Abdal Aziz,Elmoghayar, Mohamed Rifaat Hamza,Ramiz, Mahmoud Mohamed Mahfouz
, p. 65 - 68 (2007/10/02)
The substituted thioureas 3a-h, prepared from 3-phenyl-2-propenoyl isothiocyanate (1) and aromatic or heteroaromatic amines 2a-h, cyclize in the presence of sodium ethoxide to give the perhydropyrimidine derivatives 5a-c.