1050329-75-3Relevant academic research and scientific papers
Discovery of a potent, selective, and less flexible selective norepinephrine reuptake inhibitor (sNRI)
Wu, Dongpei,Pontillo, Joseph,Ching, Brett,Hudson, Sarah,Gao, Yinghong,Fleck, Beth A.,Gogas, Kathleen,Wade, Warren S.
, p. 4224 - 4227 (2008)
The design, synthesis, and SAR of a series of ring-constrained norepinephrine reuptake inhibitors are described. A substantially rigid inhibitor with potent functional activity at the transporter (IC50 = 8 nM) was used to develop a model for th
