105855-73-0Relevant articles and documents
Efficient synthesis and evaluation of bimodal ligand NETA
Chong, Hyun-Soon,Song, Hyun A.,Birch, Noah,Le, Thien,Lim, Sooyoun,Ma, Xiang
scheme or table, p. 3436 - 3439 (2009/04/11)
The efficient and short synthetic route to the structurally novel bimodal ligand NETA for antibody-targeted radiation therapy (radioimmunotherapy, RIT) of cancer was developed. The structure of NETA was determined by X-ray crystallography. The arsenazo-ba
Scorpionate-like pendant macrocyclic ligands, complexes and compositions thereof, and methods of using same
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Page 9, (2008/06/13)
Substituted 1,4,7-triazacyclononane-N,N′,N″-triacetic acid compounds with a pendant donor amino group, metal complexes thereof, compositions thereof, and methods of use in diagnostic imaging and treatment of a cellular disorder.
Synthesis and biological evaluation of novel macrocyclic ligands with pendent donor groups as potential yttrium chelators for radioimmunotherapy with improved complex formation kinetics
Chong, Hyun-Soon,Garmestani, Kayhan,Ma, Dangshe,Milenic, Diane E.,Overstreet, Terrish,Brechbiel, Martin W.
, p. 3458 - 3464 (2007/10/03)
Novel 1,4,7-triazacyclononane-N,N′,N″-triacetic acid (NOTA) based octadentate ligands [2-(4,7-biscarboxymethyl[1,4,7]triazacyclononan-1- ylethyl)carbonylmethylamino] acetic acid tetrahydrochloride (1) and [3-(4,7-biscarboxymethyl[1,4,7]triazacyclononan-1-
Macrobicyclic Amonoethers with Twelve-membered Rings
Alfheim, Tore,Buoeen, Solfrid,Dale, Johannes,Krautwurst, Klaus D.
, p. 40 - 49 (2007/10/02)
A one-pot reaction between alkane-1,2-diamines and triethyleneglycol ditosylate, or similar compounds having tosylamine functions instead of ether functions, gives without high dilution good yields of bicyclic compounds consisting of two twelve-membered rings with the alkane-diamine unit in common.The simplest representatives, 4,7,13,16-tetraoxa-1,10-diaza-bicycloeicosane and its 19-substituted derivatives, show strong cation complexation with a high selectivity for Na+ over Li+ and K+.Dynamic NMR spectroscopy shows that confomational processes, including amine inversion, are fast when the ethylene bridge is unsubstituted but become hindered when a methyl substituent is present.