1061214-81-0Relevant articles and documents
Design, synthesis, and structure-affinity relationship studies in NK1 receptor ligands based on azole-fused quinolinecarboxamide moieties
Cappelli, Andrea,Giuliani, Germano,Anzini, Maurizio,Riitano, Daniela,Giorgi, Gianluca,Vomero, Salvatore
, p. 6850 - 6859 (2008)
The substituent in position 2 of the quinoline nucleus of NK1 receptor ligands 5 has been constrained into different five-membered heterocyclic moieties in order to obtain information on the binding site pocket interacting with this apparently
HETEROTRICYCLIC AMIDE DERIVATIVES AS NEUROKININ-l (NKl) RECEPTOR LIGANDS
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Page/Page column 7; 12, (2010/11/27)
The present invention relates to compounds of formula 1, method of preparation and uses thereof.