1070798-64-9Relevant academic research and scientific papers
Synthesis and calpain inhibitory activity of peptidomimetic compounds with constrained amino acids at the P2 position
Donkor, Isaac O.,Korukonda, Rajani
, p. 4806 - 4808 (2008)
The effect of incorporating α,α′-diethylglycine and α-aminocyclopentane carboxylic acid at the P2 position of inhibitors on μ-calpain inhibition was studied. Compound 3 with α,α′-diethylglycine was over 20-fold more potent than 2 with α-aminocy
