1073340-44-9Relevant academic research and scientific papers
Synthesis and evaluation of structurally constrained quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists
Nagase, Tsuyoshi,Mizutani, Takashi,Sekino, Etsuko,Ishikawa, Shiho,Ito, Sayaka,Mitobe, Yuko,Miyamoto, Yasuhisa,Yoshimoto, Ryo,Tanaka, Takeshi,Ishihara, Akane,Takenaga, Norihiro,Tokita, Shigeru,Sato, Nagaaki
experimental part, p. 6889 - 6901 (2009/10/23)
A series of structurally constrained derivatives of the potent H 3 inverse agonist 1 was designed, synthesized, and evaluated as histamine H3 receptor inverse agonists. As a result, the N-cyclobutylpiperidin-4-yloxy group as in 2f wa
