1079084-08-4Relevant academic research and scientific papers
Design and synthesis of fluorescent SGLT2 inhibitors
Lansdell, Mark I.,Burring, Denise J.,Hepworth, David,Strawbridge, Matthew,Graham, Emily,Guyot, Thierry,Betson, Mark S.,Hart, James D.
scheme or table, p. 4944 - 4947 (2009/05/07)
The design and synthesis of the first fluorophore-conjugated SGLT2 inhibitors is described. The mode of linking the fluorophore to the SGLT2 pharmacophore was found to be crucial in achieving optimum potency. Superior potency to phlorizin was provided by
