1079396-24-9Relevant articles and documents
Imidazole derivative and application thereof as TRPV4 inhibitor
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Paragraph 0071-0072, (2020/10/29)
The invention relates to imidazole derivatives of formula (I) and pharmaceutically acceptable salts, isomers, prodrugs and pharmaceutical compositions thereof. The compounds are inhibitors of vanilloid 4 type transient receptor potential channels (TRPV4).
BICYCLIC HETEROCYCLE DERIVATIVES AND THEIR USE AS GPCR MODULATORS
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Page/Page column 53, (2010/04/03)
The present invention relates to Bicyclic Heterocycle Derivatives of Formula (I), compositions comprising a Bicyclic Heterocycle Derivative, and methods of using the Bicyclic Heterocycle Derivatives for treating or preventing obesity, diabetes, a diabetic
[6,5]-BICYCLIC GPR119 G PROTEIN-COUPLED RECEPTOR AGONISTS
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Page/Page column 70-71, (2009/01/20)
Novel compounds are provided which are GPR119 G protein-coupled receptor modulators. GPR119 G protein-coupled receptor modulators are useful in treating, preventing, or slowing the progression of diseases requiring GPR119 G protein-coupled receptor modulator therapy. These novel compounds have the structure: or stereoisomers or prodrugs or pharmaceutically acceptable salts thereof, wherein n2, n3, n4, A, B, D, E, G, J, Y, R1 and R2 are defined herein.