108445-06-3Relevant academic research and scientific papers
Arylaminoethyl amides as novel non-covalent cathepsin K inhibitors
Altmann, Eva,Renaud, Johanne,Green, Jonathan,Farley, David,Cutting, Brian,Jahnke, Wolfgang
, p. 2352 - 2354 (2007/10/03)
A series of Nα-benzyloxycarbonyl- and Nα-acyl-L-leucine(2-phenylaminoethyl)amide derivatives were prepared and evaluated for their inhibitory activity against rabbit and human cysteine proteases cathepsins K, L, and S. These data ind
SYNTHESIS OF 1,2-AMINOAZIDES. CONVERSION TO UNSYMMETRICAL VICINAL DIAMINES BY CATALYTIC HYDROGENATION OR REDUCTIVE ALKYLATION WITH DICHLOROBORANES.
Benalil, Aziza,Carboni, Bertrand,Vaultier, Michel
, p. 8177 - 8194 (2007/10/02)
1,2-aminoazides are easily prepared from 1,2-amino alcohols.Catalytic hydrogenation in the presence of palladium on charcoal or reductive alkylation with dichloroboranes afford with good yields unsymmetrically substituted vicinal diamines.
A CONVENIENT SYNTHESIS OF N-ARYL-N'-BENZYL-1,2-ETHANEDIAMINES
Lis, Randall,Marisca, Anthony J.
, p. 45 - 50 (2007/10/02)
A practical and convenient synthesis of N-Aryl-N'-benzyl-1,2-ethanediamines 5-10 from various anilines and N-benzyl-2-chloroethylamine hydrochloride is described.
