1092545-65-7Relevant articles and documents
Synthesis and SAR of analogs of the M1 allosteric agonist TBPB. Part II: Amides, sulfonamides and ureas-The effect of capping the distal basic piperidine nitrogen
Miller, Nicole R.,Daniels, R. Nathan,Bridges, Thomas M.,Brady, Ashley E.,Conn, P. Jeffrey,Lindsley, Craig W.
scheme or table, p. 5443 - 5447 (2009/05/30)
This letter describes the further synthesis and SAR, developed through an iterative analog library approach, of analogs of the highly selective M1 allosteric agonist TBPB by deletion of the distal basic piperidine nitrogen by the formation of amides, sulf