1094780-13-8Relevant articles and documents
Highly potent 4-amino-indolo[2,3-c]azepin-3-one-containing somatostatin mimetics with a range of sst receptor selectivities
Feytens, Debby,De Vlaeminck, Magali,Cescato, Renzo,Tourwé, Dirk,Reubi, Jean Claude
experimental part, p. 95 - 104 (2009/08/09)
The synthesis, biological evaluation, and conformational analysis of 4-amino-indolo[2,3-c]azepin-3-one (Aia)- containing SRIF mimetics are reported. Different subtype selectivities are observed depending on the N- and C-terminal substituents of the D-Aia-