111627-48-6Relevant articles and documents
SYNTHESIS PROCESS, AND CRYSTALLINE FORM OF 4-BENZAMIDE HYDROCHLORIDE AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT
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Page/Page column 4, (2013/02/27)
Industrial synthesis process for, and crystalline form I of, the compound of formula (I): and also crystalline form I of the associated free base. Medicinal products containing the same which are useful in the treatment of disorders of the histaminergic system.
Acetamide scanning around bicyclic thiazoles: SAR at the H3 receptor
Denonne, Frederic,Celanire, Sylvain,Christophe, Bernard,Defays, Sabine,Delaunoy, Christel,Delporte, Marie-Laure,Detrait, Eric,Durieu, Veronique,Gillard, Michel,Lamberty, Yves,Lorent, Genevieve,Nicolas, Jean-Marie,van Bellinghen, Alain,van Houtvin, Nathalie,Provins, Laurent
scheme or table, p. 1559 - 1565 (2012/01/06)
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Phenyl-oxazoles, a new family of inverse agonists at the H3 histamine receptor
Denonne, Frederic,Atienzar, Franck,Celanire, Sylvain,Christophe, Bernard,Delannois, Frederique,Delaunoy, Christel,Delporte, Marie-Laure,Durieu, Vronique,Gillard, Michel,Lallemand, Bndicte,Lamberty, Yves,Lorent, Genevive,Vanbellinghen, Alain,Van Houtvin, Nathalie,Verbois, Valrie,Provins, Laurent
scheme or table, p. 206 - 212 (2010/12/24)
(Chemical Equation Presented) Drug design: Oxazoles and thiazoles were designed and synthesised based on previously reported ligands of the 3rd histamine receptor (H3R). The aminopropoxy-phenyl-oxazole chemotype was identified as a promising H