1126530-07-1Relevant academic research and scientific papers
Synthesis and conformation#activity relationships of the peptide isosteres of FK228 and largazole
Bowers, Albert A.,Greshook, Thomas J.,West, Nathan,Estiu, Guillermina,Schreiber, Stuart L.,et al.
supporting information; experimental part, p. 2900 - 2905 (2009/07/30)
The peptide isosteres (10 and 11) of the naturally occurring and potent histone deacetylase (HDAC) Inhibitors FK228 and largazole have been synthesized and evaluated side-by-side with FK228, largazole, and SAHA for inhibition of the class I HDACs 1, 2, 3,
