1128075-68-2Relevant academic research and scientific papers
Site-selective azaindole arylation at the azine and azole rings via N-oxide activation
Huestis, Malcolm P.,Fagnou, Keith
supporting information; experimental part, p. 1357 - 1360 (2009/09/05)
Subjection of N-methyl 6-and 7-azaindole N-oxides to a Pd(OAc) 2/DavePhos catalyst system enables regioselective direct arylation of the azine ring. Following deoxygenation, 7-azaindole substrates undergo an additional regioselective azole direct arylation event in good yield.
