112811-91-3Relevant academic research and scientific papers
A convenient synthesis of n-substituted 2,3-dihydro-3-oxoisothiazolo[5,4-b]pyridines in acidic conditions
Terauchi, Hideo,Tanitame, Akihiko,Tada, Keiko,Nishikawa, Yoshinori
, p. 1719 - 1734 (2007/10/03)
A novel and convenient synthesis of N-substituted 2,3-dihydro-3-oxoisothiazolo[5,4-b]pyridines which possess potent in vitro inhibitory activity against gastric (H+/K+)-ATPase is reported. Compared with the methods reported previously, the compounds were synthesized more readily in relatively high yields by conversion of N-substituted 2-(benzyl-, 1-phenylethyl-, and benzhydrylsulfinyl)nicotinamides (17d-l) in a diluted hydrochloric acid-methanol solution at room temperature.
Herbicidal o-carbomethoxy-sulfonylureas
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, (2008/06/13)
The compound 2-[[(4,6-dimethoxypyrimidin-2-yl)amino-carbonyl]-aminosulfonyl]-3-pyridinecarboxylic acid, methyl ester is useful as an agricultural chemical. It has high herbicidal activity, desirable spectrum of weed control and low residual activity. As s
