114380-33-5Relevant academic research and scientific papers
Atroposelective Haloamidation of Indoles with Amino Acid Derivatives and Hypohalides
Li, Zhaojie,Tang, Menghan,Hu, Chenyang,Yu, Shouyun
, p. 8819 - 8823 (2019)
An atroposelective coupling of indoles with chiral amino acid-based sulfonamides mediated by hypohalides is described. A series of 2-amido-3-haloindoles with a C-N chiral axis are delivered using this strategy. The C3 halogen atoms can facilitate further
Controllable synthesis of 3-chloro- and 3,3-dichloro-2-oxindoles via hypervalent iodine-mediated chlorooxidation
Jiang, Xinpeng,Yang, Liechao,Yang, Wenlong,Zhu, Yu,Fang, Liyun,Yu, Chuanming
, p. 6920 - 6924 (2019)
An efficient and controllable protocol for the synthesis of 3-chloro- and 3,3-dichloro-2-oxindoles has been developed via hypervalent iodine-promoted chlorooxidation. By using two equivalents of 1-chloro-1,2-benziodoxol-3-(1H)-one, a wide range of indoles
